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Intermediates

S/N Product Name CAS Classification
Available Intermediates
1 1,2,3-tris-o-acetyl-5-deoxy-β-D-furribose 62211-93-2 Capecitabine Intermediate
2 2′,3′-Di-O-acetyl-5′-deoxy-5-fluorocytidine 161599-46-8 Capecitabine Intermediate
3 5′-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine-2′,3′-diacetate 162204-20-8 Capecitabine Intermediate
4 N-methyl-1-naphthalenemethylamine 14489-75-9 Terbinafine Hydrochloride Intermediate
5 N-Methyl-1-Naphthalenemethylamine Hydrochloride 65473-13-4 Terbinafine Hydrochloride Intermediate
6 3,3-Dimethyl-1-Butyne 917-92-0 Terbinafine Hydrochloride Intermediate
7 1-chloro-6,6-dimethyl-2-hepten-4-yne 126764-17-8 Terbinafine Hydrochloride Intermediate
8 4-(4-Fluorobenzoyl)butyric acid 149437-76-3 Ezetimibe Intermediate
9 (4S)-3-[5-(4-Fluorophenyl)-1,5-dioxopenyl]-4-phenyl-2-oxazolidinone 189028-93-1 Ezetimibe Intermediate
10 (4S)-3-[(5S)-5-(4-fluorophenyl)-5-hydroxypentanoyl]-4-phenyl-1,3-oxazolidin-2-one 189028-95-3 Ezetimibe Intermediate
11 4-[[(4-Fluorophenyl)imino]methyl]-phenol 3382-63-6 Ezetimibe Intermediate
12 3-[(2R,5S)-5-(4-Fluorophenyl)-2-[(S)-[(4-fluorophenyl(amino)]][4-[trimethylsilyl]-oxy]phenyl]methyl]-1-oxo-5-[(trimethylsily)-oxy]pentyl]-4-phenyl-(4S)-2-oxazolidinone 272778-12-8 Ezetimibe Intermediate
13 Cis-Hexahydroisoindoline 1470-99-1 Mitiglinide Calcium Intermediate
14 Cis-Hexahydroisoindoline Hydrochloride 161829-92-1 Mitiglinide Calcium Intermediate
15 2-Benzylsuccinic Acid 36092-42-9 Mitiglinide Calcium Intermediate
16 (S)-2-Benzylsuccinic Acid 3972-36-9 Mitiglinide Calcium Intermediate
17 2-BenzylAcrylic Acid 5669-19-2 Racecadotril Intermediate
18 Benzyl glycinate p-toluenesulfonate 1738-76-7 Racecadotril Intermediate
19 2-[(Acetylthio)methyl]-3-phenylpropionic Acid 91702-98-6 Racecadotril Intermediate
20 3-Chloro-1-(3-fluorobenzyloxy)-4-nitrobenzene 443882-99-3 Lapatinib Intermediate
21 3-Chloro-4-(3-fluorobenzyloxy)aniline 202197-26-0 Lapatinib Intermediate
22 N-[3-Chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amine 231278-20-9 Lapatinib Intermediate
23 5-[4-[3-Chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-carbaldehyde 231278-84-5 Lapatinib Intermediate
24 6-Iodoquinazolin-4-one 16064-08-7 Lapatinib Intermediate
25 4-Chloro-6-iodoquinazoline 98556-31-1 Lapatinib Intermediate
26 5-Formylfuran-2-boronic acid 27329-70-0 Lapatinib Intermediate
27 2-(Methylsulfonyl)ethylamine Hydrochloride 104458-24-4 Lapatinib Intermediate
28 Methyl 7-Methoxy-4-oxo-1,4-dihydroquinoline-6-carboxylate 205448-65-3 Lenvatinib Intermediate
29 4-Amino-3-chlorophenol 17609-80-2 Lenvatinib Intermediate
30 4-Amino-3-chlorophenol Hydrochloride 52671-64-4 Lenvatinib Intermediate
31 Methyl 4-chloro-7-Methoxyquinoline-6-carboxylate 205448-66-4 Lenvatinib Intermediate
32 4-Chloro-7-methoxyquinoline-6-carboxamide 417721-36-9 Lenvatinib Intermediate
33 1-(2-chloro-4-hydroxyphenyl)-3-cyclopropylurea 796848-79-8 Lenvatinib Intermediate
34 2-amino-5-bromopyridine 1072-97-5 Palbociclib Intermediate
35 2,4-Dichloropyrimidine 3934-20-1 Palbociclib Intermediate
36 5-Bromo-2,4-dichloropyrimidine 36082-50-5 Palbociclib Intermediate
37 5-Bromo-2-nitropyridine 39856-50-3 Palbociclib Intermediate
38 4-(6-Nitro-3-pyridyl)-piperazine-1-carboxylate 571189-16-7 Palbociclib Intermediate
39 tert-Butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate 571188-59-5 Palbociclib Intermediate
40 5-broMo-2-chloro-N-cyclopentylpyriMidin-4-aMine 733039-20-8 Palbociclib Intermediate
41 2-Chloro-8-Cyclopentyl-5-Methyl Pyrido[2,3-d]Pyrimidin-7(8h)-One 1013916-37-4 Palbociclib Intermediate
42 6-Bromo-2-chloro-8-cyclopentyl-5-methylpyrido-[2,3-d]pyrimidin-7(8H)-one 1016636-76-2 Palbociclib Intermediate
43 4-{6-[(6-bromo-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino)]-pyridin-3-yl}-piperazine-1-carboxylic acid-butyl ester 571188-82-4 Palbociclib Intermediate
44 tert-butyl 4-(6-(8-cyclopentyl-5-Methyl-7-oxo-6-(1-propoxyvinyl)-7,8-dihydropyrido[2,3-d]pyriMidin-2-ylaMino)pyridin-3-yl)piperazine-1-carboxylate 866084-31-3 Palbociclib Intermediate
45 2-chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyriMidine-6-carboxylic acid 1211443-58-1 Ribociclib Intermediate
46 2-Chloro-7-cyclopentyl-7H-cyclopentyl[d]pyrimidin-6-carboxamide 1211443-61-6 Ribociclib Intermediate
47 3-(2-Chloro-4-(cyclopentylamino)pyrimidin-5-yl)prop-2-yn-1-ol 1374639-76-5 Ribociclib Intermediate
48 (2-chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)methanol 1374639-77-6 Ribociclib Intermediate
49 2-chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidine-6-carbaldehyde 1211443-55-8 Ribociclib Intermediate
50 1-Aminocyclobutanecarboxylic acid 22264-50-2 Apalutamide Intermediate
51 5-Amino-3-(trifluoromethyl)picolinonitrile 573762-62-6 Apalutamide Intermediate
52 5-isothiocyanato-3-(trifluoromethyl)picolinonitrile 951753-87-0 Apalutamide Intermediate
53 1-((3-fluoro-4-(methylcarbamoyl)phenyl)amino)cyclobutanecarboxylic acid 2227589-22-0 Apalutamide Intermediate
54 5-Nitro-3-trifluoromethylpyridine-2-carbonitrile 573762-57-9 Apalutamide Intermediate
55 1-(Cyclopropylcarbonyl)piperazine 59878-57-8 Olaparib Intermediate
56 1-(cyclopropylcarbonyl)piperazine hydrochloride 1021298-67-8 Olaparib Intermediate
57 3-oxo-1,3-dihydroisobenzofuran-1-ylphosphonic acid 61260-15-9 Olaparib Intermediate
58 2-Fluoro-5-[(3-oxo-1(3H)-isobenzofuranylidene)methyl]-benzonitrile 763114-25-6 Olaparib Intermediate
59 2-Fluoro-5-[(4-oxo-3,4-dihydrophthalazin-1-yl)Methyl]benzoic acid 763114-26-7 Olaparib Intermediate
60 2-Fluoro-5-formylbenzonitrile 218301-22-5 Olaparib Intermediate
61 2-Fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)Methyl)benzonitrile 1021298-68-9 Olaparib Intermediate
62 2-Methyl-2-propanyl 4-{2-fluoro-5-[(4-oxo-3,4-dihydro-1-phthalazi nyl)methyl]benzoyl}-1-piperazinecarboxylate 763114-04-1 Olaparib Intermediate
63 1-[5-[(3,4-Dihydro-4-oxo-1-phthalazinyl)methyl]-2-fluorobenzoyl]piperazine 763111-47-3 Olaparib Intermediate
64 tert-butyl 4-(cyclopropanecarbonyl)piperazine-1-carboxylate 414910-15-9 Olaparib Intermediate
65 Ethyl 2-aminothiazole-5-carboxylate 32955-21-8 Dasatinib Intermediate
66 2-Amino-N-(2-chloro-6-methylphenyl)thiazole-5-carboxamide 302964-24-5 Dasatinib Intermediate
67 N-(2-Chloro-6-methylphenyl)-2-[(6-chloro-2-methyl-4-pyrimidinyl)amino]-5-thiazolecarboxamide 302964-08-5 Dasatinib Intermediate
68 2-((tert-Butoxycarbonyl)amino)thiazole-5-carboxylicacid 302964-02-9 Dasatinib Intermediate
69 4,6-Dichloro-2-methylpyrimidine 1780-26-3 Dasatinib Intermediate
70 (1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methylbutane-1-boronate 179324-87-9 Bortezomib Intermediate
71 N-(2-Pyrazinylcarbonyl)-L-phenylalanine 114457-94-2 Bortezomib Intermediate
72 N-(2′,6′-Dimethylphenyl)-2-Piperidinecarboxamide 15883-20-2 Ropivacaine Intermediate
73 (S)-N-(2′,6′-Dimethylphenyl)-2-Piperidinecarboxamide 27262-40-4 Ropivacaine Intermediate
74 (±)2,6-Diamino-4,5,6,7-tetrahydro-benzothiazole (PX-III) 104617-49-4 Pramipexole Intermediate
75 (6S)-2,6-Diamino-4,5,6,7-tetrahydro-benzothiazole 106092-09-5 Pramipexole Intermediate
76 5-Bromo-3-((trimethylsilyl)ethynyl)pyrazin-2-amine 875781-41-2 Upadacitinib Intermediate
77 2-Bromo-5-tosyl-5H-pyrrolo[2,3-b]pyrazine 1201186-54-0 Upadacitinib Intermediate
78 Carbamic acid,N-[5-[(4-methylphenyl)sulfonyl]-5H-pyrrolo[2,3-b]pyrazin-2-yl]-,ethyl este 1869118-24-0 Upadacitinib Intermediate
79 tert-butyl 5-tosyl-5H-pyrrolo[2,3-b]pyrazin-2-ylcarbamate 1201187-44-1 Upadacitinib Intermediate
80 (3R,4S)-3-(2-Bromoacetyl)-4-ethyl-1-pyrrolidinecarboxylic acid phenylmethyl ester 1428243-26-8 Upadacitinib Intermediate
81 Benzyl (3r,4s)-3-(N-(Ethoxycarbonyl)-N-(5-Tosyl-5h-Pyrrolo[2,3-B]Pyrazin-2-Yl)Glycyl)-4-Ethylpyrrolidine-1-Carboxylate 2050038-81-6 Upadacitinib Intermediate
82 benzyl (3R,4S)-3-(N-(tert-butoxycarbonyl)-N-(5-tosyl-5H-pyrrolo[2,3-b]pyrazin-2-yl)glycyl)-4-ethylpyrrolidine-1-carboxylate 1428243-27-9 Upadacitinib Intermediate
83 8-[(3R,4S)-4-ethyl-3-pyrrolidinyl]-3H-Imidazo[1,2-a]pyrrolo[2,3-e]pyrazine hydrochloride 2050038-84-9 Upadacitinib Intermediate
84 1-((Benzyloxy)carbonyl)-4-ethyl-2,5-dihydro-1H-pyrrole-3-carboxylic acid 1869118-25-1 Upadacitinib Intermediate
85 5-(2-Fluorophenyl)-1H-pyrrole-3-carboxaldehyde 881674-56-2 Vonoprazan Intermediate
86 3-pyridylsulfonyl chloride 16133-25-8 Vonoprazan Intermediate
87 1H-Pyrrole-3-carboxaldehyde, 5-(2-fluorophenyl)-1-(3-pyridinylsulfonyl)- 881677-11-8 Vonoprazan Intermediate
88 [2-(2-fluorophenyl)-2-oxoethyl]propanedinitrile 312307-38-3 Vonoprazan Intermediate
89 5-(2-Fluorophenyl)-1H-pyrrole-3-carbonitrile 1240948-77-9 Vonoprazan Intermediate
90 Diethyl 1,3-acetonedicarboxylate 105-50-0 Strontium Ranelate Intermediate
91 5-amino-4-cyano-3-(2-ethoxy-2-oxoethyl)thiophene-2-carboxylate 58168-20-0 Strontium Ranelate Intermediate
92 Tetraethyl Ranelate 58194-26-6 Strontium Ranelate Intermediate
93 2,3-Pyridinedicarboxylic acid dimethyl ester 605-38-9 Rimegepant Intermediate
94 dimethyl 5,9-dihydroxy-7H-cyclohepta[b]pyridine-6,8-dicarboxylate 39713-36-5 Rimegepant Intermediate
95 7,8-Dihydro-5H-cyclohepta[b]pyridine-5,9(6H)-dione 39713-40-1 Rimegepant Intermediate
96 (R)-9-((triisopropylsilyl)oxy)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-5-onehydrochloride 1190363-45-1 Rimegepant Intermediate
97 (6S,9R)-6-(2,3-Difluorophenyl)-6,7,8,9-tetrahydro-9-[[tris(1-methylethyl)silyl]oxy]-5H-cyclohepta[b]pyridin-5-one 1190363-46-2 Rimegepant Intermediate
98 (5S,6S,9R)-6-(2,3-difluorophenyl)-9-((triisopropylsilyl)oxy)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-5-aminedihydrochloride 1373116-04-1 Rimegepant Intermediate
99 2,​3-​Pyridinediamine-N3-​4-​piperidinyl-​dihydrochloride 1373116-08-5 Rimegepant Intermediate
100 1-(1-(1H-imidazole-1-carbonyl)piperidin-4-yl)-1H-imidazo[4,5-b]pyridin-2(3H)-one 1373116-06-3 Rimegepant Intermediate
101 (5S,6S,9R)-5-amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-ol:dihydrochloride 1373116-07-4 Rimegepant Intermediate
102 ethyl-2,2-dimethyl-7-bromoheptanoate 123469-92-1 Bempedoic Acid Intermediate
103 2,2,14,14-tetramethyl-8-oxopentadecanedioic acid diethyl ester 738606-43-4 Bempedoic Acid Intermediate
104 2,2,14,14-tetramethyl-8-oxopentadecanedioic acid 413624-71-2 Bempedoic Acid Intermediate

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